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Masitinib is a broad coronavirus 3CL inhibitor that blocks replication of SARS-CoV-2 期刊论文
Science, 2021
作者:  Nir Drayman;  Jennifer K. DeMarco;  Krysten A. Jones;  Saara-Anne Azizi;  Heather M. Froggatt;  Kemin Tan;  Natalia Ivanovna Maltseva;  Siquan Chen;  Vlad Nicolaescu;  Steve Dvorkin;  Kevin Furlong;  Rahul S. Kathayat;  Mason R. Firpo;  Vincent Mastrodomenico;  Emily A. Bruce;  Madaline M. Schmidt;  Robert Jedrzejczak;  Miguel Á. Muñoz-Alía;  Brooke Schuster;  Vishnu Nair;  Kyu-yeon Han;  Amornrat O’Brien;  Anastasia Tomatsidou;  Bjoern Meyer;  Marco Vignuzzi;  Dominique Missiakas;  Jason W. Botten;  Christopher B. Brooke;  Hyun Lee;  Susan C. Baker;  Bryan C. Mounce;  Nicholas S. Heaton;  William E. Severson;  Kenneth E. Palmer;  Bryan C. Dickinson;  Andrzej Joachimiak;  Glenn Randall;  Savaş Tay
收藏  |  浏览/下载:13/0  |  提交时间:2021/08/25
Heterogeneity of meningeal B cells reveals a lymphopoietic niche at the CNS borders 期刊论文
Science, 2021
作者:  Simone Brioschi;  Wei-Le Wang;  Vincent Peng;  Meng Wang;  Irina Shchukina;  Zev J. Greenberg;  Jennifer K. Bando;  Natalia Jaeger;  Rafael S. Czepielewski;  Amanda Swain;  Denis A. Mogilenko;  Wandy L. Beatty;  Peter Bayguinov;  James A. J. Fitzpatrick;  Laura G. Schuettpelz;  Catrina C. Fronick;  Igor Smirnov;  Jonathan Kipnis;  Virginia S. Shapiro;  Gregory F. Wu;  Susan Gilfillan;  Marina Cella;  Maxim N. Artyomov;  Steven H. Kleinstein;  Marco Colonna
收藏  |  浏览/下载:22/0  |  提交时间:2021/07/27
Revealing x-ray and gamma ray temporal and spectral similarities in the GRB 190829A afterglow 期刊论文
Science, 2021
作者:  H.E.S.S. Collaboration;  H. Abdalla;  F. Aharonian;  F. Ait Benkhali;  E. O. Angüner;  C. Arcaro;  C. Armand;  T. Armstrong;  H. Ashkar;  M. Backes;  V. Baghmanyan;  V. Barbosa Martins;  A. Barnacka;  M. Barnard;  Y. Becherini;  D. Berge;  K. Bernlöhr;  B. Bi;  E. Bissaldi;  M. Böttcher;  C. Boisson;  J. Bolmont;  M. de Bony de Lavergne;  M. Breuhaus;  F. Brun;  P. Brun;  M. Bryan;  M. Büchele;  T. Bulik;  T. Bylund;  S. Caroff;  A. Carosi;  S. Casanova;  T. Chand;  S. Chandra;  A. Chen;  G. Cotter;  M. Curyło;  J. Damascene Mbarubucyeye;  I. D. Davids;  J. Davies;  C. Deil;  J. Devin;  L. Dirson;  A. Djannati-Ataï;  A. Dmytriiev;  A. Donath;  V. Doroshenko;  L. Dreyer;  C. Duffy;  J. Dyks;  K. Egberts;  F. Eichhorn;  S. Einecke;  G. Emery;  J.-P. Ernenwein;  K. Feijen;  S. Fegan;  A. Fiasson;  G. Fichet de Clairfontaine;  G. Fontaine;  S. Funk;  M. Füßling;  S. Gabici;  Y. A. Gallant;  G. Giavitto;  L. Giunti;  D. Glawion;  J. F. Glicenstein;  M.-H. Grondin;  J. Hahn;  M. Haupt;  G. Hermann;  J. A. Hinton;  W. Hofmann;  C. Hoischen;  T. L. Holch;  M. Holler;  M. Hörbe;  D. Horns;  D. Huber;  M. Jamrozy;  D. Jankowsky;  F. Jankowsky;  A. Jardin-Blicq;  V. Joshi;  I. Jung-Richardt;  E. Kasai;  M. A. Kastendieck;  K. Katarzyński;  U. Katz;  D. Khangulyan;  B. Khélifi;  S. Klepser;  W. Kluźniak;  Nu. Komin;  R. Konno;  K. Kosack;  D. Kostunin;  M. Kreter;  G. Lamanna;  A. Lemière;  M. Lemoine-Goumard;  J.-P. Lenain;  F. Leuschner;  C. Levy;  T. Lohse;  I. Lypova;  J. Mackey;  J. Majumdar;  D. Malyshev;  D. Malyshev;  V. Marandon;  P. Marchegiani;  A. Marcowith;  A. Mares;  G. Martí-Devesa;  R. Marx;  G. Maurin;  P. J. Meintjes;  M. Meyer;  A. Mitchell;  R. Moderski;  L. Mohrmann;  A. Montanari;  C. Moore;  P. Morris;  E. Moulin;  J. Muller;  T. Murach;  K. Nakashima;  A. Nayerhoda;  M. de Naurois;  H. Ndiyavala;  J. Niemiec;  L. Oakes;  P. O’Brien;  H. Odaka;  S. Ohm;  L. Olivera-Nieto;  E. de Ona Wilhelmi;  M. Ostrowski;  S. Panny;  M. Panter;  R. D. Parsons;  G. Peron;  B. Peyaud;  Q. Piel;  S. Pita;  V. Poireau;  A. Priyana Noel;  D. A. Prokhorov;  H. Prokoph;  G. Pühlhofer;  M. Punch;  A. Quirrenbach;  S. Raab;  R. Rauth;  P. Reichherzer;  A. Reimer;  O. Reimer;  Q. Remy;  M. Renaud;  F. Rieger;  L. Rinchiuso;  C. Romoli;  G. Rowell;  B. Rudak;  E. Ruiz-Velasco;  V. Sahakian;  S. Sailer;  H. Salzmann;  D. A. Sanchez;  A. Santangelo;  M. Sasaki;  M. Scalici;  J. Schäfer;  F. Schüssler;  H. M. Schutte;  U. Schwanke;  M. Seglar-Arroyo;  M. Senniappan;  A. S. Seyffert;  N. Shafi;  J. N. S. Shapopi;  K. Shiningayamwe;  R. Simoni;  A. Sinha;  H. Sol;  A. Specovius;  S. Spencer;  M. Spir-Jacob;  Ł. Stawarz;  L. Sun;  R. Steenkamp;  C. Stegmann;  S. Steinmassl;  C. Steppa;  T. Takahashi;  T. Tam;  T. Tavernier;  A. M. Taylor;  R. Terrier;  J. H. E. Thiersen;  D. Tiziani;  M. Tluczykont;  L. Tomankova;  M. Tsirou;  R. Tuffs;  Y. Uchiyama;  D. J. van der Walt;  C. van Eldik;  C. van Rensburg;  B. van Soelen;  G. Vasileiadis;  J. Veh;  C. Venter;  P. Vincent;  J. Vink;  H. J. Völk;  Z. Wadiasingh;  S. J. Wagner;  J. Watson;  F. Werner;  R. White;  A. Wierzcholska;  Yu Wun Wong;  A. Yusafzai;  M. Zacharias;  R. Zanin;  D. Zargaryan;  A. A. Zdziarski;  A. Zech;  S. J. Zhu;  J. Zorn;  S. Zouari;  N. Żywucka;  P. Evans;  K. Page
收藏  |  浏览/下载:36/0  |  提交时间:2021/06/15
Dynamic remodeling of host membranes by self-organizing bacterial effectors 期刊论文
Science, 2021
作者:  Ting-Sung Hsieh;  Victor A. Lopez;  Miles H. Black;  Adam Osinski;  Krzysztof Pawłowski;  Diana R. Tomchick;  Jen Liou;  Vincent S. Tagliabracci
收藏  |  浏览/下载:9/0  |  提交时间:2021/06/07
X-ray screening identifies active site and allosteric inhibitors of SARS-CoV-2 main protease 期刊论文
Science, 2021
作者:  Sebastian Günther;  Patrick Y. A. Reinke;  Yaiza Fernández-García;  Julia Lieske;  Thomas J. Lane;  Helen M. Ginn;  Faisal H. M. Koua;  Christiane Ehrt;  Wiebke Ewert;  Dominik Oberthuer;  Oleksandr Yefanov;  Susanne Meier;  Kristina Lorenzen;  Boris Krichel;  Janine-Denise Kopicki;  Luca Gelisio;  Wolfgang Brehm;  Ilona Dunkel;  Brandon Seychell;  Henry Gieseler;  Brenna Norton-Baker;  Beatriz Escudero-Pérez;  Martin Domaracky;  Sofiane Saouane;  Alexandra Tolstikova;  Thomas A. White;  Anna Hänle;  Michael Groessler;  Holger Fleckenstein;  Fabian Trost;  Marina Galchenkova;  Yaroslav Gevorkov;  Chufeng Li;  Salah Awel;  Ariana Peck;  Miriam Barthelmess;  Frank Schlünzen;  P. Lourdu Xavier;  Nadine Werner;  Hina Andaleeb;  Najeeb Ullah;  Sven Falke;  Vasundara Srinivasan;  Bruno Alves França;  Martin Schwinzer;  Hévila Brognaro;  Cromarte Rogers;  Diogo Melo;  Joanna J. Zaitseva-Doyle;  Juraj Knoska;  Gisel E. Peña-Murillo;  Aida Rahmani Mashhour;  Vincent Hennicke;  Pontus Fischer;  Johanna Hakanpää;  Jan Meyer;  Philip Gribbon;  Bernhard Ellinger;  Maria Kuzikov;  Markus Wolf;  Andrea R. Beccari;  Gleb Bourenkov;  David von Stetten;  Guillaume Pompidor;  Isabel Bento;  Saravanan Panneerselvam;  Ivars Karpics;  Thomas R. Schneider;  Maria Marta Garcia-Alai;  Stephan Niebling;  Christian Günther;  Christina Schmidt;  Robin Schubert;  Huijong Han;  Juliane Boger;  Diana C. F. Monteiro;  Linlin Zhang;  Xinyuanyuan Sun;  Jonathan Pletzer-Zelgert;  Jan Wollenhaupt;  Christian G. Feiler;  Manfred S. Weiss;  Eike-Christian Schulz;  Pedram Mehrabi;  Katarina Karničar;  Aleksandra Usenik;  Jure Loboda;  Henning Tidow;  Ashwin Chari;  Rolf Hilgenfeld;  Charlotte Uetrecht;  Russell Cox;  Andrea Zaliani;  Tobias Beck;  Matthias Rarey;  Stephan Günther;  Dusan Turk;  Winfried Hinrichs;  Henry N. Chapman;  Arwen R. Pearson;  Christian Betzel;  Alke Meents
收藏  |  浏览/下载:14/0  |  提交时间:2021/05/14
Aberrant type 1 immunity drives susceptibility to mucosal fungal infections 期刊论文
Science, 2021
作者:  Timothy J. Break;  Vasileios Oikonomou;  Nicolas Dutzan;  Jigar V. Desai;  Marc Swidergall;  Tilo Freiwald;  Daniel Chauss;  Oliver J. Harrison;  Julie Alejo;  Drake W. Williams;  Stefania Pittaluga;  Chyi-Chia R. Lee;  Nicolas Bouladoux;  Muthulekha Swamydas;  Kevin W. Hoffman;  Teresa Greenwell-Wild;  Vincent M. Bruno;  Lindsey B. Rosen;  Wint Lwin;  Andy Renteria;  Sergio M. Pontejo;  John P. Shannon;  Ian A. Myles;  Peter Olbrich;  Elise M. N. Ferré;  Monica Schmitt;  Daniel Martin;  Genomics and Computational Biology Core16;  Daniel L. Barber;  Norma V. Solis;  Luigi D. Notarangelo;  David V. Serreze;  Mitsuru Matsumoto;  Heather D. Hickman;  Philip M. Murphy;  Mark S. Anderson;  Jean K. Lim;  Steven M. Holland;  Scott G. Filler;  Behdad Afzali;  Yasmine Belkaid;  Niki M. Moutsopoulos;  Michail S. Lionakis
收藏  |  浏览/下载:13/0  |  提交时间:2021/01/22
Enteroviral 3C protease activates the human NLRP1 inflammasome in airway epithelia 期刊论文
Science, 2020
作者:  Kim S. Robinson;  Daniel Eng Thiam Teo;  Kai Sen Tan;  Gee Ann Toh;  Hsiao Hui Ong;  Chrissie Kaishi Lim;  Kenneth Lay;  Bijin Veonice Au;  Tian Sheng Lew;  Justin Jang Hann Chu;  Vincent Tak Kwong Chow;  De Yun Wang;  Franklin L. Zhong;  Bruno Reversade
收藏  |  浏览/下载:6/0  |  提交时间:2020/12/07
Capturing roaming molecular fragments in real time 期刊论文
Science, 2020
作者:  Tomoyuki Endo;  Simon P. Neville;  Vincent Wanie;  Samuel Beaulieu;  Chen Qu;  Jude Deschamps;  Philippe Lassonde;  Bruno E. Schmidt;  Hikaru Fujise;  Mizuho Fushitani;  Akiyoshi Hishikawa;  Paul L. Houston;  Joel M. Bowman;  Michael S. Schuurman;  François Légaré;  Heide Ibrahim
收藏  |  浏览/下载:9/0  |  提交时间:2020/11/30
Patterning and growth control in vivo by an engineered GFP gradient 期刊论文
Science, 2020
作者:  Kristina S. Stapornwongkul;  Marc de Gennes;  Luca Cocconi;  Guillaume Salbreux;  Jean-Paul Vincent
收藏  |  浏览/下载:2/0  |  提交时间:2020/10/20
Antitumor activity of a systemic STING-activating non-nucleotide cGAMP mimetic 期刊论文
Science, 2020
作者:  Emily N. Chin;  Chenguang Yu;  Vincent F. Vartabedian;  Ying Jia;  Manoj Kumar;  Ana M. Gamo;  William Vernier;  Sabrina H. Ali;  Mildred Kissai;  Daniel C. Lazar;  Nhan Nguyen;  Laura E. Pereira;  Brent Benish;  Ashley K. Woods;  Sean B. Joseph;  Alan Chu;  Kristen A. Johnson;  Philipp N. Sander;  Francisco Martínez-Peña;  Eric N. Hampton;  Travis S. Young;  Dennis W. Wolan;  Arnab K. Chatterjee;  Peter G. Schultz;  H. Michael Petrassi;  John R. Teijaro;  Luke L. Lairson
收藏  |  浏览/下载:19/0  |  提交时间:2020/08/25